NVP 231

CAS No. 362003-83-6

NVP 231 ( NVP231; NVP 231; NVP-231 )

Catalog No. M14241 CAS No. 362003-83-6

NVP-231 is a potent, specific, and reversible CerK inhibitor(IC50=12±2 nM) that competitively inhibits binding of ceramide to CerK.

Purity : >98%(HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 27 In Stock
10MG 43 In Stock
25MG 70 In Stock
50MG 113 In Stock
100MG 186 In Stock
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Biological Information

  • Product Name
    NVP 231
  • Note
    Research use only, not for human use.
  • Brief Description
    NVP-231 is a potent, specific, and reversible CerK inhibitor(IC50=12±2 nM) that competitively inhibits binding of ceramide to CerK.
  • Description
    NVP-231 is a potent, specific, and reversible CerK inhibitor(IC50=12±2 nM) that competitively inhibits binding of ceramide to CerK.
  • Synonyms
    NVP231; NVP 231; NVP-231
  • Pathway
    MAPK/ERK Signaling
  • Target
    ERK
  • Recptor
    CERK
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    362003-83-6
  • Formula Weight
    431.55
  • Molecular Formula
    C25H25N3O2S
  • Purity
    >98%(HPLC)
  • Solubility
    Soluble in DMSO
  • SMILES
    O=C(C1(C2)C[C@H]3C[C@@H]2C[C@H](C3)C1)NC4=CC=C5N=C(NC(C6=CC=CC=C6)=O)SC5=C4
  • Chemical Name
    N -[2-(Benzoylamino)-6-benzothiazolyl]tricyclo[3.3.1.13,7]decane-1-carboxamide

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Graf C, et al.Mol Pharmacol. 2008 Oct;74(4):925-32.
molnova catalog
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